This webinar takes place on Thursday September 18th between 16.00 and 16.45 CEST / 15.00-15.45 BST / 10.00-10.45 AM EST / 7.00-7.45 AM PST.
Follow the link to register for the webinar. Please note that the presentation will be given during the live event only and on demand viewing at a later date will not be possible. Contact us for any questions.
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Abstract:
Human genomic approaches are identifying more and more genes that are associated with chronic pain. For many of these genes, the physiological association to chronic pain is not self-evident. Furthermore, methods to efficiently validate such targets functionally are currently lacking.
In this webinar, we will glance at Orion’s approach for identification and prioritization of genetically associated pain targets in their Drug Discovery programs. Furthermore, we will present how the combination of lentiviral knock-down (KD) and high-capacity electrophysiology could be used to functionally validate pain targets. In the latter part, we will share data from a proof-of-concept (PoC) study where neuronal excitability (a key hallmark of pain) was evaluated after KD of genetically linked pain targets, e.g. Nav1.7. After the positive outcome of the PoC, the methodology was applied to screen novel pain targets. We will end by discussing how the outcome aided in enabling Orion to rank and prioritize between these targets.